List of Protease Inhibitors

Code Product Target Protease Package
3165-v Ac-Tyr-Val-Ala-Asp-H (aldehyde) [Ac-YVAD-CHO] Caspase-1 5 mg
3166-v Ac-Tyr-Val-Lys-Asp-H (aldehyde) [Ac-YVKD-CHO] Caspase-1 5 mg
3169-v Z-Ile-Glu(OBut)-Ala-Leu-H (aldehyde) [PSI] Proteasome 5 mg
3170-v Z-Leu-Leu-Nva-H (aldehyde) [MG-115] Proteasome 5 mg
3172-v Ac-Asp-Glu-Val-Asp-H (aldehyde) [Ac-DEVD-CHO] Caspase-3/7/8 5 mg
3173-v Biotinyl-Asp-Glu-Val-Asp-H (aldehyde) [Biot-DEVD-CHO] Caspase-3/7/8 1 mg
3174-v Z-Asp-CH2-DCB Caspases 5 mg
3175-v Z-Leu-Leu-Leu-H (aldehyde) [MG-132] Proteasome and Cathepsin K 5 mg
3178-v Z-Leu-Leu-H (aldehyde) Calpain 5 mg
3180-v Ac-Tyr-Val-Ala-Asp-CH2Cl [Ac-YVAD-CMK] Caspases 5 mg
3182-v Ac-Val-Glu-Ile-Asp-H (aldehyde) [Ac-VEID-CHO] Caspase-6 5 mg
3187-v Ac-Trp-Glu-His-Asp-H (aldehyde) [Ac-WEHD-CHO] Caspase-1 5 mg
3188-v Z-Val-Ala-Asp(OMe)-CH2F [Z-VAD-FMK] Caspases 1 mg
3192-v Ac-Asp-Met-Gln-Asp-H (aldehyde) [Ac-DMQD-CHO] Caspase-3 5 mg
3194-v Ac-Asp-Gln-Thr-Asp-H (aldehyde) [Ac-DQTD-CHO] Caspase-7/3 5 mg
3196-v Ac-Ile-Glu-Thr-Asp-H (aldehyde) [Ac-IETD-CHO] Caspase-8/6 and Granzyme B 5 mg
3199-v Ac-Leu-Glu-His-Asp-H (aldehyde) [Ac-LEHD-CHO] Caspase-9 5 mg
3202-v Ala-Ala-Phe-CH2Cl [AAF-CMK] Tripeptidyl Peptidase II, Chymotrypsin, and Chymase 5 mg
3204-v Ac-Val-Asp-Val-Ala-Asp-H (aldehyde) [Ac-VDVAD-CHO] Caspase-2 5 mg
3207-v Ubiquitin Aldehyde Deubiquitinating Enzyme 50 μg
3214-v SUAM-14746 Prolyl Endopeptidase 5 mg
3218-v (Z-Leu-Leu-NHCH2)2CO [(Z-LL)2 Ketone] Signal Peptide Peptidase 5 mg
3219-v (3,5-Difluorophenylacetyl)-Ala-Phg-OBut
[DAPT]
γ-Secretase 5 mg
3221-v Ac-Asp-Asn-Leu-Asp-H (aldehyde)
[Ac-DNLD-CHO]
Caspase-3 5 mg
3223-v Bz-Arg-His-D-Asp-CH2Cl [Bz-RHd-CMK] D-Aspartyl Endopeptidase 5 mg
3241-v Ac-Lys-Val-Pro-Leu-CH2Cl [Ac-KVPL-CMK] Granzyme M 5 mg
3253-v Ac-Abu-D-Tyr-Leu-Gln-VS SARS-CoV-2 Main Protease 1 mg
3254-v Boc-Asp(OMe)-CH2F [Boc-D-FMK] Caspases 5 mg
4041 Leupeptin Trypsin, Plasmin, Papain and Cathepsin B 25 mg
100 mg
1 g
4041-v Leupeptin Trypsin, Plasmin, Papain and Cathepsin B 0.5 mg
4062 Antipain Trypsin, u-PA, Papain and Cathepsin A/B 25 mg
100 mg
4062-v Antipain Trypsin, u-PA, Papain and Cathepsin A/B 0.5 mg
4063 Chymostatin Chymotrypsin, Chymase, Papain and Cathepsin B/G 25 mg
100 mg
4063-v Chymostatin Chymotrypsin, Chymase, Papain and Cathepsin B/G 0.5 mg
4064 Elastatinal Elastase 25 mg
100 mg
4064-v Elastatinal Elastase 0.5 mg
4082 Phosphoramidon Thermolysin and Endothelin Converting Enzyme 25 mg
100 mg
4082-v Phosphoramidon Thermolysin and Endothelin Converting Enzyme 0.5 mg
4095 Amastatin Aminopeptidase A/PS and Leucyl Aminopeptidase 25 mg
4095-v Amastatin Aminopeptidase A/PS and Leucyl Aminopeptidase 0.5 mg
4096 E-64 Thiol Proteases 25 mg
100 mg
1 g
4096-v E-64 Thiol Proteases 0.5 mg
4132 Diprotin A Dipeptidyl-Aminopeptidase IV 25 mg
100 mg
4146 Cl-Ac-(OH)Leu-Ala-Gly-NH2 Elastase 25 mg
100 mg
4149 Arphamenine B Aminopeptidase B 25 mg
100 mg
4149-v Arphamenine B Aminopeptidase B 0.5 mg
4155 Ebelactone A N-Formylmethionine Aminopeptidase 25 mg
4320-v E-64-c Cathepsin B/H/L and Calpain 5 mg
4321-v E-64-d Cathepsin B/H/L and Calpain 5 mg
4322-v CA-074 Cathepsin B 5 mg
4323-v CA-074 Me Cathepsin B 5 mg
4342-v Phebestin Aminopeptidase N 5 mg
4368-v Lactacystin Proteasome 0.2 mg
4378-v Lys-Thr-Glu-Glu-Ile-Ser-Glu-Val-Asn-Sta-Val-Ala-Glu-Phe β-Secretase/td>

1 mg
4381-v Epoxomicin Proteasome 0.2 mg
4394-v L-685,458 γ-Secretase 1 mg
4395-v KYT-1 Arg-Gingipain 1 mg
4396-v KYT-36 Lys-Gingipain/td>

1 mg
4397 Pepstatin A Pepsin, Cathepsin D/E and Renin 25 mg
100 mg
1 g
4397-v Pepstatin A Pepsin, Cathepsin D/E and Renin 0.5 mg
4519 Ile-Pro-Pro [IPP] ACE1 100 mg
4520 Val-Pro-Pro [VPP] ACE1 100 mg
4523-v KYT-41 Arg-Gingipain and Lys-Gingipain 1 mg


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