[Pyr1]-Apelin-13 (Human)

Code:
4361-v
Name:
[Pyr1]-Apelin-13 (Human)
Pyr-Arg-Pro-Arg-Leu-Ser-His-Lys-Gly-Pro-Met-Pro-Phe
(M.W. 1533.8) C69H108N22O16S
Ligand for APJ Receptor
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Vial 0.5 mg 7,000 Ships within
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Purity:
≧98.0% (HPLC)
View Analytical Data Sheet
Storage:
-20 ℃
Source:
Bovine, Rat
Production:
Synthetic Product

Solubility: H2O (0.1 mM)

more information

Category:
Biologically Active Peptides

reference

  1. K. Tatemoto, M. Hosoya, Y. Habata, R. Fujii, T. Takegawa, M.-X. Zou, Y. Kawamata, S. Fukusumi, S. Hinuma, C. Kitada, T. Kurokawa, H. Onda, and M. Fujino, Biochem. Biophys. Res. Commun., 251, 471 (1998). (Original)
  2. M.-X. Zou, H.-Y. Liu, Y. Haraguchi, Y. Soda, K. Tatemoto, and H. Hoshino, FEBS Lett., 473, 15 (2000). (Pharmacol.)
  3. M. Hosoya, Y. Kawamata, S. Fukusumi, R. Fujii, Y. Habata, S. Hinuma, C. Kitada, S. Honda, T. Kurokawa, H. Onda, O. Nishimura, and M. Fujino, J. Biol. Chem., 275, 21061 (2000). (Pharmacol.)
  4. D.K. Lee, R. Cheng, T. Nguyen, T. Fan, A.P. Kariyawasam, Y. Liu, D.H. Osmond, S.R. George, and B.F.O'Dowd, J. Neurochem., 74, 34 (2000). (cDNA Seq.; Rat)
  5. N. De Mota, A.R.-L. Goazigo, S.E. Messari, N. Chartrel, D. Roesch, C. Dujardin, C. Kordon, H. Vaudry, F. Moos, and C. Llorens-Cortes, Proc. Natl. Acad. Sci. U.S.A., 101, 10464 (2004). (Endogenous Apelin 13 in Rat)
  6. S.C. Sorli, L. van den Berghe, B. Masri, B. Knibiehler, and Y. Audigier, Drug Discov. Today, 11, 1100 (2006). (Review)
  7. C. Carpene, C. Dray, C. Attane, P. Valet, M.P. Portillo, I. Churruca, F.I. Milagro, and I. Castan-Laure, J. Physiol. Biochem.,, 63, 359 (2007). (Review)
  8. I. Falcao-Pires, R. Ladeiras-Lopes, and A.F. Leite-Moreira, Expert Opin. Ther. Targets, 14, 633 (2010). (Review)

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