4095 Amastatin

Code:
4095
Name:
Amastatin
[(2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-L-valyl-L-valyl-L-aspartic acid
(M.W. 474.55) C21H38N4O8
Inhibitor for Aminopeptidase A/PS and Leucyl Aminopeptidase
Package Price(Yen)
Bulk 25 mg 99,300

main

Purity:
≧98.0% (HPLC)
Other Name:
アマスタチン
Storage:
-20 ℃
Production:
Synthetic Product

more information

Structure:
structure of Amastatin
CAS Registry Number:
67655-94-1
Category:
Enzyme Inhibitors

reference

  1. T. Aoyagi, H. Tobe, F. Kojima, M. Hamada, T. Takeuchi, and H. Umezawa, J. Antibiotics, 31, 636 (1978). (Original)
  2. H. Tobe, H. Morishima, H. Naganawa, T. Takita, T. Aoyagi, and H. Umezawa, Agric. Biol. Chem., 43, 591 (1979). (Structure & Chem. Synthesis)
  3. P.M. Dando and A.J. Barrett, In, Enzyme 343. Aminopeptidase PS, Handbook of Proteolytic Enzymes, (A.J. Barrett, N.D. Rawlings, and J.F. Woessner eds.), Academic Press, New York, (1998). (Inhibitory Activity)
  4. D. Leung, G. Abbenante, and D.P. Fairlie, J. Med. Chem., 43, 305 (2000).