4095-v Amastatin

Code:
4095-v
Name:
Amastatin
[(2S,3R)-3-Amino-2-hydroxy-5-methylhexanoyl]-L-valyl-L-valyl-L-aspartic acid
(M.W. 474.55) C21H38N4O8
Inhibitor for Aminopeptidase A/PS and Leucyl Aminopeptidase
Package Price(Yen)
Vial 0.5 mg 6,900

main

Purity:
≧98.0% (HPLC)
Other Name:
アマスタチン
Storage:
-20 ℃
Production:
Synthetic Product

Solubility: DMSO or AcOH (10 mM)

more information

Structure:
構造図Amastatin
CAS Registry Number:
67655-94-1
Category:
Enzyme Inhibitors

reference

  1. T. Aoyagi, H. Tobe, F. Kojima, M. Hamada, T. Takeuchi, and H. Umezawa, J. Antibiotics, 31, 636 (1978). (Original)
  2. H. Tobe, H. Morishima, H. Naganawa, T. Takita, T. Aoyagi, and H. Umezawa, Agric. Biol. Chem., 43, 591 (1979). (Structure & Chem. Synthesis)
  3. P.M. Dando and A.J. Barrett, In, Enzyme 343. Aminopeptidase PS, Handbook of Proteolytic Enzymes, (A.J. Barrett, N.D. Rawlings, and J.F. Woessner eds.), Academic Press, New York, (1998). (Inhibitory Activity)
  4. D. Leung, G. Abbenante, and D.P. Fairlie, J. Med. Chem., 43, 305 (2000).