3219-v (3,5-Difluorophenylacetyl)-Ala-Phg-OBut

Code:
3219-v
Name:
(3,5-Difluorophenylacetyl)-Ala-Phg-OBut
DAPT
(3,5-Difluorophenylacetyl)-L-alanyl-L-2-phenylglycine t-butyl ester
(M.W. 432.46) C23H26N2O4F2
Inhibitor for γ-Secretase
Package Price(Yen)
Vial 5 mg 10,000

main

Purity:
≧99.0% (HPLC)
Storage:
-20 ℃
Production:
Synthetic Product

Solubility: DMSO (10 mM)

more information

Structure:
構造図(3,5-Difluorophenylacetyl)-Ala-Phg-OBut
CAS Registry Number:
208255-80-5
Category:
Enzyme Inhibitors

reference

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  2. A.Y. Kornilova, C. Das, and M.S. Wolfe, J. Biol. Chem., 278, 16470 (2003). (Comparison of in Cells and Cell-Free Activity)
  3. D. Leung, G. Abbenante, and D.P. Fairlie, J. Med. Chem., 43, 305 (2000).